Saccharin as a salt former. Enhanced solubilities of saccharinates of active pharmaceutical ingredients.

نویسندگان

  • Prashant M Bhatt
  • Nittala V Ravindra
  • Rahul Banerjee
  • Gautam R Desiraju
چکیده

Saccharin, acting as a weak acid, forms salts with basic APIs and these salts have the desirable property of enhanced water solubility.

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عنوان ژورنال:
  • Chemical communications

دوره 8  شماره 

صفحات  -

تاریخ انتشار 2005